Mebhydrolin napadisylate is a specific histamine H1 receptor antagonist.

Product information

CAS Number: 6153-33-9

Molecular Weight: 841.05

Formula: C48H48N4O6S2

Chemical Name: bis(5-benzyl-2-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole); naphthalene-1,5-disulfonic acid

Smiles: CN1CC2C3C=CC=CC=3N(CC3C=CC=CC=3)C=2CC1.CN1CC2C3C=CC=CC=3N(CC3C=CC=CC=3)C=2CC1.OS(=O)(=O)C1=CC=CC2C1=CC=CC=2S(O)(=O)=O

InChiKey: CJUOSBUQOWKEKJ-UHFFFAOYSA-N

InChi: InChI=1S/2C19H20N2.C10H8O6S2/c2*1-20-12-11-19-17(14-20)16-9-5-6-10-18(16)21(19)13-15-7-3-2-4-8-15;11-17(12,13)9-5-1-3-7-8(9)4-2-6-10(7)18(14,15)16/h2*2-10H,11-14H2,1H3;1-6H,(H,11,12,13)(H,14,15,16)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : 14.29 mg/mL (16.99 mM; ultrasonic and warming and heat to 60°C).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 ^oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 ^oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vitro:

Mebhydrolin is a specific histamine H1-receptor antagonist with minimal sedative properties and comparing it with the effects of chlorpromazine, the archetypical phenothiazine. Mebhydrolin exerts an antihistaminic effect over the period of the ethanol interaction study.

Products are for research use only. Not for human use.