Cariprazine D8 (RGH-188 D8) is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

Product information

CAS Number: 1308278-50-3

Molecular Weight: 435.46

Formula: C21H32Cl2N4O

Chemical Name: 3-((1r, 4r)-4-(2-(4-(2, 3-dichlorophenyl)piperazin-1-yl-2, 2, 3, 3, 5, 5, 6, 6-d8)ethyl)cyclohexyl)-1, 1-dimethylurea

Smiles: [2H]C1([2H])N(CC[C@@H]2CC[C@H](CC2)NC(=O)N(C)C)C([2H])([2H])C([2H])([2H])N(C2=CC=CC(Cl)=C2Cl)C1([2H])[2H] |&1:6,9|

InChiKey: KPWSJANDNDDRMB-OMZDLYIGSA-N

InChi: InChI=1S/C21H32Cl2N4O/c1-25(2)21(28)24-17-8-6-16(7-9-17)10-11-26-12-14-27(15-13-26)19-5-3-4-18(22)20(19)23/h3-5,16-17H,6-15H2,1-2H3,(H,24,28)/t16-,17-/i12D2,13D2,14D2,15D2

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 ^oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 ^oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.